4SC-202 tosylate
CAS No. 1186222-89-8
4SC-202 tosylate ( 4SC-202 )
Catalog No. M17177 CAS No. 1186222-89-8
4SC-202 is a selective inhibitor of class I HDAC for HDAC1/2/3 (IC50: 1.20/1.12/0.57 μM). It also displays inhibitory activity against Lysine-specific demethylase 1 (LSD1).
Purity : 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
2MG | 53 | In Stock |
|
5MG | 87 | In Stock |
|
10MG | 132 | In Stock |
|
25MG | 240 | In Stock |
|
50MG | 399 | In Stock |
|
100MG | 588 | In Stock |
|
200MG | Get Quote | In Stock |
|
500MG | Get Quote | In Stock |
|
1G | Get Quote | In Stock |
|
Biological Information
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Product Name4SC-202 tosylate
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NoteResearch use only, not for human use.
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Brief Description4SC-202 is a selective inhibitor of class I HDAC for HDAC1/2/3 (IC50: 1.20/1.12/0.57 μM). It also displays inhibitory activity against Lysine-specific demethylase 1 (LSD1).
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Description4SC-202 is a selective inhibitor of class I HDAC for HDAC1/2/3 (IC50: 1.20/1.12/0.57 μM). It also displays inhibitory activity against Lysine-specific demethylase 1 (LSD1).
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Synonyms4SC-202
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PathwayMetabolic Enzyme/Protease
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TargetPhosphatase
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RecptorHDAC1;HDAC2;HDAC3;HDAC5;HDAC9;HDAC10;HDAC11;
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number1186222-89-8
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Formula Weight619.71
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Molecular FormulaC30H29N5O6S2
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Purity98%
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SolubilityDMSO : ≥ 51 mg/mL. 82.30 mM
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SMILESCC1=CC=C(C=C1)S(=O)(=O)O.CN1C=C(C=N1)C2=CC=C(C=C2)S(=O)(=O)N3C=CC(=C3)/C=C/C(=O)NC4=CC=CC=C4N
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Pinkerneil M, Hoffmann M J, Kohlhof H, et al. Targeted Oncology, 2016, 11(6):783-798.
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