4SC-202 tosylate

CAS No. 1186222-89-8

4SC-202 tosylate ( 4SC-202 )

Catalog No. M17177 CAS No. 1186222-89-8

4SC-202 is a selective inhibitor of class I HDAC for HDAC1/2/3 (IC50: 1.20/1.12/0.57 μM). It also displays inhibitory activity against Lysine-specific demethylase 1 (LSD1).

Purity : 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 53 In Stock
5MG 87 In Stock
10MG 132 In Stock
25MG 240 In Stock
50MG 399 In Stock
100MG 588 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    4SC-202 tosylate
  • Note
    Research use only, not for human use.
  • Brief Description
    4SC-202 is a selective inhibitor of class I HDAC for HDAC1/2/3 (IC50: 1.20/1.12/0.57 μM). It also displays inhibitory activity against Lysine-specific demethylase 1 (LSD1).
  • Description
    4SC-202 is a selective inhibitor of class I HDAC for HDAC1/2/3 (IC50: 1.20/1.12/0.57 μM). It also displays inhibitory activity against Lysine-specific demethylase 1 (LSD1).
  • Synonyms
    4SC-202
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    Phosphatase
  • Recptor
    HDAC1;HDAC2;HDAC3;HDAC5;HDAC9;HDAC10;HDAC11;
  • Research Area
    Cancer
  • Indication
    ——

Chemical Information

  • CAS Number
    1186222-89-8
  • Formula Weight
    619.71
  • Molecular Formula
    C30H29N5O6S2
  • Purity
    98%
  • Solubility
    DMSO : ≥ 51 mg/mL. 82.30 mM
  • SMILES
    CC1=CC=C(C=C1)S(=O)(=O)O.CN1C=C(C=N1)C2=CC=C(C=C2)S(=O)(=O)N3C=CC(=C3)/C=C/C(=O)NC4=CC=CC=C4N
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Pinkerneil M, Hoffmann M J, Kohlhof H, et al. Targeted Oncology, 2016, 11(6):783-798.
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